VX-680 KINOMEscan - Dataset (ID:20197)

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Small Molecule Protein Kd Conc unit
Tozasertib DAPK3 9900.0
nM
Tozasertib HUNK 9800.0
nM
Tozasertib PAK6 9700.0
nM
Tozasertib ACVRL1 9500.0
nM
Tozasertib DRAK1 9000.0
nM
Tozasertib NEK7 8700.0
nM
Tozasertib TEC 8700.0
nM
Tozasertib CHEK1 8700.0
nM
Tozasertib BRSK1 8400.0
nM
Tozasertib TGFBR1 8400.0
nM
Tozasertib TTK 8100.0
nM
Tozasertib RSK1(Kin.Dom.1-N-terminal) 7900.0
nM
Tozasertib LTK 7500.0
nM
Tozasertib FES 7400.0
nM
Tozasertib ABL1(F317I)-nonphosphorylated 7200.0
nM
Tozasertib FGFR4 7200.0
nM
Tozasertib BMPR2 7100.0
nM
Tozasertib ERBB3 7100.0
nM
Tozasertib CAMK1 7000.0
nM
Tozasertib NDR2 6900.0
nM
Tozasertib ERK5 6800.0
nM
Tozasertib TYK2(JH2domain-pseudokinase) 6600.0
nM
Tozasertib CAMK1G 6500.0
nM
Tozasertib LATS2 6500.0
nM
Tozasertib RSK2(Kin.Dom.1-N-terminal) 6400.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records