VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | DAPK3 | 9900.0 | nM |
Tozasertib | HUNK | 9800.0 | nM |
Tozasertib | PAK6 | 9700.0 | nM |
Tozasertib | ACVRL1 | 9500.0 | nM |
Tozasertib | DRAK1 | 9000.0 | nM |
Tozasertib | NEK7 | 8700.0 | nM |
Tozasertib | TEC | 8700.0 | nM |
Tozasertib | CHEK1 | 8700.0 | nM |
Tozasertib | BRSK1 | 8400.0 | nM |
Tozasertib | TGFBR1 | 8400.0 | nM |
Tozasertib | TTK | 8100.0 | nM |
Tozasertib | RSK1(Kin.Dom.1-N-terminal) | 7900.0 | nM |
Tozasertib | LTK | 7500.0 | nM |
Tozasertib | FES | 7400.0 | nM |
Tozasertib | ABL1(F317I)-nonphosphorylated | 7200.0 | nM |
Tozasertib | FGFR4 | 7200.0 | nM |
Tozasertib | BMPR2 | 7100.0 | nM |
Tozasertib | ERBB3 | 7100.0 | nM |
Tozasertib | CAMK1 | 7000.0 | nM |
Tozasertib | NDR2 | 6900.0 | nM |
Tozasertib | ERK5 | 6800.0 | nM |
Tozasertib | TYK2(JH2domain-pseudokinase) | 6600.0 | nM |
Tozasertib | CAMK1G | 6500.0 | nM |
Tozasertib | LATS2 | 6500.0 | nM |
Tozasertib | RSK2(Kin.Dom.1-N-terminal) | 6400.0 | nM |