HKI-272 KINOMEscan-2 - Dataset (ID:20195)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | MST1R | 8400.0 | nM |
| Neratinib | FAK2 | 8000.0 | nM |
| Neratinib | CSNK1G3 | 7800.0 | nM |
| Neratinib | PAK6 | 7500.0 | nM |
| Neratinib | RSK1(Kin.Dom.1-N-terminal) | 7400.0 | nM |
| Neratinib | ABL1(Q252H)-nonphosphorylated | 7100.0 | nM |
| Neratinib | MET(M1250T) | 6700.0 | nM |
| Neratinib | KC1G2 | 6600.0 | nM |
| Neratinib | YANK2 | 6400.0 | nM |
| Neratinib | FLT3(N841I) | 6400.0 | nM |
| Neratinib | RIPK5 | 6400.0 | nM |
| Neratinib | FYN | 6400.0 | nM |
| Neratinib | ABL1(Q252H)-phosphorylated | 6000.0 | nM |
| Neratinib | MLK3 | 5800.0 | nM |
| Neratinib | CHEK1 | 5700.0 | nM |
| Neratinib | CAMK1D | 5600.0 | nM |
| Neratinib | MAST1 | 5500.0 | nM |
| Neratinib | MLK1 | 5400.0 | nM |
| Neratinib | FLT3 | 5400.0 | nM |
| Neratinib | STK36 | 5300.0 | nM |
| Neratinib | SYK | 5100.0 | nM |
| Neratinib | CDK7 | 5100.0 | nM |
| Neratinib | FLT3(K663Q) | 4900.0 | nM |
| Neratinib | TXK | 4800.0 | nM |
| Neratinib | MLK2 | 4600.0 | nM |