HKI-272 KINOMEscan-2 - Dataset (ID:20195)

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Small Molecule Protein Kd Conc unit
Neratinib EGFR(G719C) 0.4
nM
Neratinib EGFR(L861Q) 0.4
nM
Neratinib EGFR(S752-I759del) 0.6
nM
Neratinib EGFR(L747-E749del, A750P) 0.6
nM
Neratinib MAP4K5 0.7
nM
Neratinib EGFR(L858R) 0.7
nM
Neratinib EGFR(G719S) 0.9
nM
Neratinib EGFR(L747-S752del, P753S) 0.9
nM
Neratinib EGFR(L747-T751del,Sins) 1.0
nM
Neratinib EGFR 1.1
nM
Neratinib EGFR(T790M) 1.5
nM
Neratinib EGFR(E746-A750del) 2.3
nM
Neratinib ERBB4 2.4
nM
Neratinib ERBB2 6.0
nM
Neratinib MST3 6.5
nM
Neratinib MST4 7.4
nM
Neratinib ERBB3 7.7
nM
Neratinib M4K3 7.7
nM
Neratinib YSK1 12.0
nM
Neratinib LOK 13.0
nM
Neratinib MP2K1 14.0
nM
Neratinib YSK4 16.0
nM
Neratinib MP2K2 26.0
nM
Neratinib EGFR(L858R,T790M) 27.0
nM
Neratinib MINK 29.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records