SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | HCK | 3.40 | nM |
Bosutinib | HIPK1 | 520.00 | nM |
Bosutinib | HIPK2 | 1900.00 | nM |
Bosutinib | HIPK3 | 3200.00 | nM |
Bosutinib | HIPK4 | 130.00 | nM |
Bosutinib | M4K1 | 15.00 | nM |
Bosutinib | HUNK | 5000.00 | nM |
Bosutinib | ICK | nM | |
Bosutinib | IGF1R | nM | |
Bosutinib | IKKA | nM | |
Bosutinib | IKKB | nM | |
Bosutinib | IKKE | 53.00 | nM |
Bosutinib | INSR | nM | |
Bosutinib | INSRR | nM | |
Bosutinib | IRAK1 | 600.00 | nM |
Bosutinib | IRAK3 | nM | |
Bosutinib | IRAK4 | 360.00 | nM |
Bosutinib | ITK | 1700.00 | nM |
Bosutinib | JAK1(JH1domain-catalytic) | nM | |
Bosutinib | JAK1(JH2domain-pseudokinase) | nM | |
Bosutinib | JAK2(JH1domain-catalytic) | 1100.00 | nM |
Bosutinib | JAK3(JH1domain-catalytic) | 1200.00 | nM |
Bosutinib | JNK1 | nM | |
Bosutinib | MK09 | nM | |
Bosutinib | JNK3 | nM |