SKI-606 KINOMEscan - Dataset (ID:20184)

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Small Molecule Protein Kd Conc unit
Bosutinib FES 330.00
nM
Bosutinib FGFR1
nM
Bosutinib FGFR2
nM
Bosutinib FGFR3
nM
Bosutinib FGFR3(G697C)
nM
Bosutinib FGFR4
nM
Bosutinib FGR 6.30
nM
Bosutinib VGFR1
nM
Bosutinib FLT3 2200.00
nM
Bosutinib FLT3(D835H) 1000.00
nM
Bosutinib FLT3(D835Y) 1100.00
nM
Bosutinib FLT3(ITD) 2900.00
nM
Bosutinib FLT3(K663Q) 2200.00
nM
Bosutinib FLT3(N841I) 3400.00
nM
Bosutinib FLT3(R834Q)
nM
Bosutinib FLT4
nM
Bosutinib FRK 1.40
nM
Bosutinib FYN 11.00
nM
Bosutinib GAK 1.30
nM
Bosutinib GCN2(Kin.Dom.2,S808G) 270.00
nM
Bosutinib GRK1
nM
Bosutinib GRK4 4900.00
nM
Bosutinib GRK7 1700.00
nM
Bosutinib GSK3A
nM
Bosutinib GSK3B
nM