SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | FES | 330.00 | nM |
Bosutinib | FGFR1 | nM | |
Bosutinib | FGFR2 | nM | |
Bosutinib | FGFR3 | nM | |
Bosutinib | FGFR3(G697C) | nM | |
Bosutinib | FGFR4 | nM | |
Bosutinib | FGR | 6.30 | nM |
Bosutinib | VGFR1 | nM | |
Bosutinib | FLT3 | 2200.00 | nM |
Bosutinib | FLT3(D835H) | 1000.00 | nM |
Bosutinib | FLT3(D835Y) | 1100.00 | nM |
Bosutinib | FLT3(ITD) | 2900.00 | nM |
Bosutinib | FLT3(K663Q) | 2200.00 | nM |
Bosutinib | FLT3(N841I) | 3400.00 | nM |
Bosutinib | FLT3(R834Q) | nM | |
Bosutinib | FLT4 | nM | |
Bosutinib | FRK | 1.40 | nM |
Bosutinib | FYN | 11.00 | nM |
Bosutinib | GAK | 1.30 | nM |
Bosutinib | GCN2(Kin.Dom.2,S808G) | 270.00 | nM |
Bosutinib | GRK1 | nM | |
Bosutinib | GRK4 | 4900.00 | nM |
Bosutinib | GRK7 | 1700.00 | nM |
Bosutinib | GSK3A | nM | |
Bosutinib | GSK3B | nM |