SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | KIT | 420.00 | nM |
Bosutinib | KIT(A829P) | 270.00 | nM |
Bosutinib | KIT(D816H) | 180.00 | nM |
Bosutinib | KIT(D816V) | 73.00 | nM |
Bosutinib | KIT(L576P) | 520.00 | nM |
Bosutinib | KIT(V559D) | 430.00 | nM |
Bosutinib | KIT(V559D,T670I) | nM | |
Bosutinib | KIT(V559D,V654A) | 130.00 | nM |
Bosutinib | LATS1 | nM | |
Bosutinib | LATS2 | nM | |
Bosutinib | LCK | 0.59 | nM |
Bosutinib | LIMK1 | nM | |
Bosutinib | LIMK2 | nM | |
Bosutinib | LKB1 | nM | |
Bosutinib | LOK | 7.00 | nM |
Bosutinib | LRRK2 | 500.00 | nM |
Bosutinib | LRRK2(G2019S) | 830.00 | nM |
Bosutinib | LTK | 3000.00 | nM |
Bosutinib | LYN | 4.20 | nM |
Bosutinib | M3K13 | 480.00 | nM |
Bosutinib | MAK | nM | |
Bosutinib | MAP3K1 | 4400.00 | nM |
Bosutinib | MAP3K15 | nM | |
Bosutinib | M3K2 | 30.00 | nM |
Bosutinib | MAP3K3 | 54.00 | nM |