BMS-540215 KINOMEscan - Dataset (ID:20180)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Brivanib | EGFR(L861Q) | 5300.0 | nM |
Brivanib | EGFR(L858R) | 5100.0 | nM |
Brivanib | ABL1(F317L)-nonphosphorylated | 4100.0 | nM |
Brivanib | KIT(D816V) | 4000.0 | nM |
Brivanib | YANK2 | 3900.0 | nM |
Brivanib | STK33 | 3200.0 | nM |
Brivanib | MP2K5 | 3100.0 | nM |
Brivanib | EGFR(G719C) | 3000.0 | nM |
Brivanib | RIPK2 | 2900.0 | nM |
Brivanib | HCK | 2700.0 | nM |
Brivanib | EGFR(G719S) | 2600.0 | nM |
Brivanib | ABL1(F317L)-phosphorylated | 2300.0 | nM |
Brivanib | BLK | 2000.0 | nM |
Brivanib | CSF1R | 1900.0 | nM |
Brivanib | ABL2 | 1800.0 | nM |
Brivanib | EPHA7 | 1700.0 | nM |
Brivanib | ABL1(T315I)-nonphosphorylated | 1700.0 | nM |
Brivanib | SRC | 1600.0 | nM |
Brivanib | ABL1(Q252H)-nonphosphorylated | 1500.0 | nM |
Brivanib | MAP4K5 | 1400.0 | nM |
Brivanib | EPHB6 | 1400.0 | nM |
Brivanib | ABL1(Q252H)-phosphorylated | 1200.0 | nM |
Brivanib | ABL1-nonphosphorylated | 1100.0 | nM |
Brivanib | TIE1 | 1100.0 | nM |
Brivanib | ABL1(Y253F)-phosphorylated | 1100.0 | nM |