BMS-540215 KINOMEscan - Dataset (ID:20180)

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Small Molecule Protein Kd Conc unit
Brivanib EGFR(L861Q) 5300.0
nM
Brivanib EGFR(L858R) 5100.0
nM
Brivanib ABL1(F317L)-nonphosphorylated 4100.0
nM
Brivanib KIT(D816V) 4000.0
nM
Brivanib YANK2 3900.0
nM
Brivanib STK33 3200.0
nM
Brivanib MP2K5 3100.0
nM
Brivanib EGFR(G719C) 3000.0
nM
Brivanib RIPK2 2900.0
nM
Brivanib HCK 2700.0
nM
Brivanib EGFR(G719S) 2600.0
nM
Brivanib ABL1(F317L)-phosphorylated 2300.0
nM
Brivanib BLK 2000.0
nM
Brivanib CSF1R 1900.0
nM
Brivanib ABL2 1800.0
nM
Brivanib EPHA7 1700.0
nM
Brivanib ABL1(T315I)-nonphosphorylated 1700.0
nM
Brivanib SRC 1600.0
nM
Brivanib ABL1(Q252H)-nonphosphorylated 1500.0
nM
Brivanib MAP4K5 1400.0
nM
Brivanib EPHB6 1400.0
nM
Brivanib ABL1(Q252H)-phosphorylated 1200.0
nM
Brivanib ABL1-nonphosphorylated 1100.0
nM
Brivanib TIE1 1100.0
nM
Brivanib ABL1(Y253F)-phosphorylated 1100.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records