BMS-540215 KINOMEscan - Dataset (ID:20180)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Brivanib | AAK1 | nM | |
Brivanib | ABL1(E255K)-phosphorylated | 580.0 | nM |
Brivanib | ABL1(F317I)-nonphosphorylated | nM | |
Brivanib | ABL1(F317I)-phosphorylated | nM | |
Brivanib | ABL1(F317L)-nonphosphorylated | 4100.0 | nM |
Brivanib | ABL1(F317L)-phosphorylated | 2300.0 | nM |
Brivanib | ABL1(H396P)-nonphosphorylated | 390.0 | nM |
Brivanib | ABL1(H396P)-phosphorylated | 640.0 | nM |
Brivanib | ABL1(M351T)-phosphorylated | 450.0 | nM |
Brivanib | ABL1(Q252H)-nonphosphorylated | 1500.0 | nM |
Brivanib | ABL1(Q252H)-phosphorylated | 1200.0 | nM |
Brivanib | ABL1(T315I)-nonphosphorylated | 1700.0 | nM |
Brivanib | ABL1(T315I)-phosphorylated | 450.0 | nM |
Brivanib | ABL1(Y253F)-phosphorylated | 1100.0 | nM |
Brivanib | ABL1-nonphosphorylated | 1100.0 | nM |
Brivanib | ABL1-phosphorylated | 640.0 | nM |
Brivanib | ABL2 | 1800.0 | nM |
Brivanib | ACVR1 | nM | |
Brivanib | ACVR1B | nM | |
Brivanib | ACVR2A | nM | |
Brivanib | ACVR2B | nM | |
Brivanib | ACVRL1 | nM | |
Brivanib | ADCK3 | nM | |
Brivanib | ADCK4 | nM | |
Brivanib | AKT1 | nM |