BMS-540215 KINOMEscan - Dataset (ID:20180)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Brivanib | VGFR2 | 5.0 | nM |
| Brivanib | VGFR1 | 10.0 | nM |
| Brivanib | PGFRA | 11.0 | nM |
| Brivanib | KIT(V559D,V654A) | 12.0 | nM |
| Brivanib | KIT(V559D,T670I) | 17.0 | nM |
| Brivanib | STK35 | 26.0 | nM |
| Brivanib | KIT(V559D) | 35.0 | nM |
| Brivanib | KIT | 36.0 | nM |
| Brivanib | PGFRB | 50.0 | nM |
| Brivanib | KIT(L576P) | 54.0 | nM |
| Brivanib | FLT4 | 56.0 | nM |
| Brivanib | FGFR1 | 99.0 | nM |
| Brivanib | FGFR2 | 110.0 | nM |
| Brivanib | FGFR3(G697C) | 150.0 | nM |
| Brivanib | TNIK | 160.0 | nM |
| Brivanib | DDR1 | 160.0 | nM |
| Brivanib | FGFR3 | 160.0 | nM |
| Brivanib | SLK | 170.0 | nM |
| Brivanib | EPHA6 | 190.0 | nM |
| Brivanib | LOK | 220.0 | nM |
| Brivanib | MINK | 310.0 | nM |
| Brivanib | RET(M918T) | 360.0 | nM |
| Brivanib | ABL1(H396P)-nonphosphorylated | 390.0 | nM |
| Brivanib | RET | 390.0 | nM |
| Brivanib | TIE2 | 440.0 | nM |