Sunitinib KINOMEscan - Dataset (ID:20179)

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Small Molecule Protein Kd Conc unit
Sunitinib KIT 0.4
nM
Sunitinib KIT(A829P) 43.0
nM
Sunitinib KIT(D816H) 110.0
nM
Sunitinib KIT(D816V) 380.0
nM
Sunitinib KIT(L576P) 1.3
nM
Sunitinib KIT(V559D) 0.4
nM
Sunitinib KIT(V559D,T670I) 0.3
nM
Sunitinib KIT(V559D,V654A) 0.2
nM
Sunitinib LATS1 630.0
nM
Sunitinib LATS2 460.0
nM
Sunitinib LCK 230.0
nM
Sunitinib LIMK1
nM
Sunitinib LIMK2
nM
Sunitinib LKB1 38.0
nM
Sunitinib LOK 19.0
nM
Sunitinib LRRK2 110.0
nM
Sunitinib LRRK2(G2019S) 76.0
nM
Sunitinib LTK 1800.0
nM
Sunitinib LYN 270.0
nM
Sunitinib M3K13 95.0
nM
Sunitinib MAK
nM
Sunitinib MAP3K1
nM
Sunitinib MAP3K15 1300.0
nM
Sunitinib M3K2 57.0
nM
Sunitinib MAP3K3 220.0
nM