Sunitinib KINOMEscan - Dataset (ID:20179)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sunitinib | KIT | 0.4 | nM |
Sunitinib | KIT(A829P) | 43.0 | nM |
Sunitinib | KIT(D816H) | 110.0 | nM |
Sunitinib | KIT(D816V) | 380.0 | nM |
Sunitinib | KIT(L576P) | 1.3 | nM |
Sunitinib | KIT(V559D) | 0.4 | nM |
Sunitinib | KIT(V559D,T670I) | 0.3 | nM |
Sunitinib | KIT(V559D,V654A) | 0.2 | nM |
Sunitinib | LATS1 | 630.0 | nM |
Sunitinib | LATS2 | 460.0 | nM |
Sunitinib | LCK | 230.0 | nM |
Sunitinib | LIMK1 | nM | |
Sunitinib | LIMK2 | nM | |
Sunitinib | LKB1 | 38.0 | nM |
Sunitinib | LOK | 19.0 | nM |
Sunitinib | LRRK2 | 110.0 | nM |
Sunitinib | LRRK2(G2019S) | 76.0 | nM |
Sunitinib | LTK | 1800.0 | nM |
Sunitinib | LYN | 270.0 | nM |
Sunitinib | M3K13 | 95.0 | nM |
Sunitinib | MAK | nM | |
Sunitinib | MAP3K1 | nM | |
Sunitinib | MAP3K15 | 1300.0 | nM |
Sunitinib | M3K2 | 57.0 | nM |
Sunitinib | MAP3K3 | 220.0 | nM |