Sunitinib KINOMEscan - Dataset (ID:20179)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sunitinib | HCK | 880.0 | nM |
Sunitinib | HIPK1 | 55.0 | nM |
Sunitinib | HIPK2 | 31.0 | nM |
Sunitinib | HIPK3 | 41.0 | nM |
Sunitinib | HIPK4 | 160.0 | nM |
Sunitinib | M4K1 | 16.0 | nM |
Sunitinib | HUNK | 500.0 | nM |
Sunitinib | ICK | 470.0 | nM |
Sunitinib | IGF1R | 2600.0 | nM |
Sunitinib | IKKA | 520.0 | nM |
Sunitinib | IKKB | nM | |
Sunitinib | IKKE | 620.0 | nM |
Sunitinib | INSR | 500.0 | nM |
Sunitinib | INSRR | 430.0 | nM |
Sunitinib | IRAK1 | 14.0 | nM |
Sunitinib | IRAK3 | 940.0 | nM |
Sunitinib | IRAK4 | 66.0 | nM |
Sunitinib | ITK | 13.0 | nM |
Sunitinib | JAK1(JH1domain-catalytic) | 6000.0 | nM |
Sunitinib | JAK1(JH2domain-pseudokinase) | 49.0 | nM |
Sunitinib | JAK2(JH1domain-catalytic) | 410.0 | nM |
Sunitinib | JAK3(JH1domain-catalytic) | 1200.0 | nM |
Sunitinib | JNK1 | nM | |
Sunitinib | MK09 | 2400.0 | nM |
Sunitinib | JNK3 | 4300.0 | nM |