TG-101348 KINOMEscan - Dataset (ID:20174)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Fedratinib | DCAMKL2 | 870.0 | nM |
| Fedratinib | DCAMKL3 | 13.0 | nM |
| Fedratinib | DDR1 | 1900.0 | nM |
| Fedratinib | DDR2 | 950.0 | nM |
| Fedratinib | M3K12 | 6300.0 | nM |
| Fedratinib | DMPK | 1000.0 | nM |
| Fedratinib | DMPK2 | nM | |
| Fedratinib | DRAK1 | 610.0 | nM |
| Fedratinib | DRAK2 | 45.0 | nM |
| Fedratinib | DYRK1A | nM | |
| Fedratinib | DYRK1B | 9500.0 | nM |
| Fedratinib | DYRK2 | nM | |
| Fedratinib | EGFR | 3400.0 | nM |
| Fedratinib | EGFR(E746-A750del) | 6200.0 | nM |
| Fedratinib | EGFR(G719C) | nM | |
| Fedratinib | EGFR(G719S) | nM | |
| Fedratinib | EGFR(L747-E749del, A750P) | 1500.0 | nM |
| Fedratinib | EGFR(L747-S752del, P753S) | 5600.0 | nM |
| Fedratinib | EGFR(L747-T751del,Sins) | 3800.0 | nM |
| Fedratinib | EGFR(L858R) | 3300.0 | nM |
| Fedratinib | EGFR(L858R,T790M) | 570.0 | nM |
| Fedratinib | EGFR(L861Q) | 5800.0 | nM |
| Fedratinib | EGFR(S752-I759del) | nM | |
| Fedratinib | EGFR(T790M) | 580.0 | nM |
| Fedratinib | EIF2AK1 | 1000.0 | nM |