TG-101348 KINOMEscan - Dataset (ID:20174)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Fedratinib | PRKX | nM | |
| Fedratinib | PRP4 | 390.0 | nM |
| Fedratinib | FAK2 | 220.0 | nM |
| Fedratinib | SIK3 | 1900.0 | nM |
| Fedratinib | RAF1 | nM | |
| Fedratinib | RET | 130.0 | nM |
| Fedratinib | RET(M918T) | 150.0 | nM |
| Fedratinib | RET(V804L) | 71.0 | nM |
| Fedratinib | RET(V804M) | 81.0 | nM |
| Fedratinib | RIOK1 | 100.0 | nM |
| Fedratinib | RIOK2 | 2600.0 | nM |
| Fedratinib | RIOK3 | 91.0 | nM |
| Fedratinib | RIPK1 | 5300.0 | nM |
| Fedratinib | RIPK2 | 6100.0 | nM |
| Fedratinib | RIPK4 | 9800.0 | nM |
| Fedratinib | RIPK5 | 1700.0 | nM |
| Fedratinib | ROCK1 | 2100.0 | nM |
| Fedratinib | ROCK2 | 2200.0 | nM |
| Fedratinib | ROS1 | 600.0 | nM |
| Fedratinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
| Fedratinib | RPS6KA4(Kin.Dom.2-C-terminal) | 140.0 | nM |
| Fedratinib | RPS6KA5(Kin.Dom.1-N-terminal) | 4400.0 | nM |
| Fedratinib | RPS6KA5(Kin.Dom.2-C-terminal) | 2200.0 | nM |
| Fedratinib | RSK1(Kin.Dom.1-N-terminal) | 1200.0 | nM |
| Fedratinib | RSK1(Kin.Dom.2-C-terminal) | 420.0 | nM |