TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib CAMK1 1600.0
nM
Fedratinib CAMK1D 460.0
nM
Fedratinib CAMK1G 3200.0
nM
Fedratinib CAMK2A 300.0
nM
Fedratinib CAMK2B 6800.0
nM
Fedratinib KCC2D 590.0
nM
Fedratinib CAMK2G 540.0
nM
Fedratinib KCC4
nM
Fedratinib KKCC1 1800.0
nM
Fedratinib CAMKK2 4000.0
nM
Fedratinib CASK 2800.0
nM
Fedratinib CDC2L1
nM
Fedratinib CDC2L2
nM
Fedratinib CDC2L5
nM
Fedratinib CDK11
nM
Fedratinib CDK2
nM
Fedratinib CDK3
nM
Fedratinib CDK4-cyclinD1 5000.0
nM
Fedratinib CDK4-cyclinD3 870.0
nM
Fedratinib CDK5
nM
Fedratinib CDK7 120.0
nM
Fedratinib CDK8
nM
Fedratinib CDK9 8800.0
nM
Fedratinib CDKL1
nM
Fedratinib CDKL2 1300.0
nM