TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib AKT2
nM
Fedratinib AKT3
nM
Fedratinib ALK 650.0
nM
Fedratinib AMPK-alpha1 2400.0
nM
Fedratinib AMPK-alpha2 4700.0
nM
Fedratinib ANKK1 4300.0
nM
Fedratinib NUAK1 34.0
nM
Fedratinib M3K5
nM
Fedratinib M3K6
nM
Fedratinib AURKA 4400.0
nM
Fedratinib AURKB 490.0
nM
Fedratinib AURKC 350.0
nM
Fedratinib AXL 160.0
nM
Fedratinib BIKE 32.0
nM
Fedratinib BLK 650.0
nM
Fedratinib BMPR1A
nM
Fedratinib BMPR1B 410.0
nM
Fedratinib BMPR2 2900.0
nM
Fedratinib BMX 1200.0
nM
Fedratinib BRAF 9800.0
nM
Fedratinib BRAF(V600E) 9300.0
nM
Fedratinib PTK6 1200.0
nM
Fedratinib BRSK1
nM
Fedratinib BRSK2
nM
Fedratinib BTK 850.0
nM