INCB018424 KINOMEscan - Dataset (ID:20173)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | JAK2(JH1domain-catalytic) | 0.0 | nM |
Ruxolitinib | TYK2(JH1domain-catalytic) | 0.9 | nM |
Ruxolitinib | JAK3(JH1domain-catalytic) | 2.0 | nM |
Ruxolitinib | JAK1(JH1domain-catalytic) | 3.4 | nM |
Ruxolitinib | M3K2 | 41.0 | nM |
Ruxolitinib | CAMK2A | 46.0 | nM |
Ruxolitinib | ROCK2 | 52.0 | nM |
Ruxolitinib | ROCK1 | 60.0 | nM |
Ruxolitinib | DCLK1 | 68.0 | nM |
Ruxolitinib | DAPK1 | 72.0 | nM |
Ruxolitinib | DAPK3 | 89.0 | nM |
Ruxolitinib | KCC2D | 90.0 | nM |
Ruxolitinib | LRRK2(G2019S) | 90.0 | nM |
Ruxolitinib | DAPK2 | 97.0 | nM |
Ruxolitinib | GAK | 99.0 | nM |
Ruxolitinib | CAMK2G | 100.0 | nM |
Ruxolitinib | CAMK1D | 120.0 | nM |
Ruxolitinib | RSK1(Kin.Dom.2-C-terminal) | 120.0 | nM |
Ruxolitinib | AAK1 | 120.0 | nM |
Ruxolitinib | PLK1 | 130.0 | nM |
Ruxolitinib | RPS6KA5(Kin.Dom.2-C-terminal) | 140.0 | nM |
Ruxolitinib | RSK4(Kin.Dom.2-C-terminal) | 150.0 | nM |
Ruxolitinib | RSK3(Kin.Dom.2-C-terminal) | 150.0 | nM |
Ruxolitinib | MAP3K3 | 150.0 | nM |
Ruxolitinib | RET(V804M) | 190.0 | nM |