INCB018424 KINOMEscan - Dataset (ID:20173)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Ruxolitinib | AAK1 | 120.0 | nM |
| Ruxolitinib | ABL1(E255K)-phosphorylated | 2200.0 | nM |
| Ruxolitinib | ABL1(F317I)-nonphosphorylated | nM | |
| Ruxolitinib | ABL1(F317I)-phosphorylated | nM | |
| Ruxolitinib | ABL1(F317L)-nonphosphorylated | 9500.0 | nM |
| Ruxolitinib | ABL1(F317L)-phosphorylated | 2200.0 | nM |
| Ruxolitinib | ABL1(H396P)-nonphosphorylated | 1100.0 | nM |
| Ruxolitinib | ABL1(H396P)-phosphorylated | nM | |
| Ruxolitinib | ABL1(M351T)-phosphorylated | 6200.0 | nM |
| Ruxolitinib | ABL1(Q252H)-nonphosphorylated | 2000.0 | nM |
| Ruxolitinib | ABL1(Q252H)-phosphorylated | 3500.0 | nM |
| Ruxolitinib | ABL1(T315I)-nonphosphorylated | nM | |
| Ruxolitinib | ABL1(T315I)-phosphorylated | nM | |
| Ruxolitinib | ABL1(Y253F)-phosphorylated | nM | |
| Ruxolitinib | ABL1-nonphosphorylated | 3700.0 | nM |
| Ruxolitinib | ABL1-phosphorylated | nM | |
| Ruxolitinib | ABL2 | nM | |
| Ruxolitinib | ACVR1 | nM | |
| Ruxolitinib | ACVR1B | nM | |
| Ruxolitinib | ACVR2A | nM | |
| Ruxolitinib | ACVR2B | nM | |
| Ruxolitinib | ACVRL1 | nM | |
| Ruxolitinib | ADCK3 | nM | |
| Ruxolitinib | ADCK4 | nM | |
| Ruxolitinib | AKT1 | nM |