INCB018424 KINOMEscan - Dataset (ID:20173)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Ruxolitinib | ABL1(F317L)-nonphosphorylated | 9500.0 | nM |
| Ruxolitinib | AURKC | 8700.0 | nM |
| Ruxolitinib | KIT(D816V) | 7100.0 | nM |
| Ruxolitinib | KIT(D816H) | 6300.0 | nM |
| Ruxolitinib | YSK1 | 6300.0 | nM |
| Ruxolitinib | KIT(A829P) | 6300.0 | nM |
| Ruxolitinib | DRAK1 | 6200.0 | nM |
| Ruxolitinib | ABL1(M351T)-phosphorylated | 6200.0 | nM |
| Ruxolitinib | EPHA3 | 6100.0 | nM |
| Ruxolitinib | GRK4 | 6100.0 | nM |
| Ruxolitinib | SgK110 | 5800.0 | nM |
| Ruxolitinib | PHKG1 | 5700.0 | nM |
| Ruxolitinib | NEK7 | 4900.0 | nM |
| Ruxolitinib | JNK1 | 4800.0 | nM |
| Ruxolitinib | CSNK2A1 | 4200.0 | nM |
| Ruxolitinib | PKNB(M.tuberculosis) | 4200.0 | nM |
| Ruxolitinib | BRAF(V600E) | 4200.0 | nM |
| Ruxolitinib | MAP3K1 | 4200.0 | nM |
| Ruxolitinib | VRK2 | 4000.0 | nM |
| Ruxolitinib | MP2K2 | 4000.0 | nM |
| Ruxolitinib | ABL1-nonphosphorylated | 3700.0 | nM |
| Ruxolitinib | DYRK2 | 3700.0 | nM |
| Ruxolitinib | ABL1(Q252H)-phosphorylated | 3500.0 | nM |
| Ruxolitinib | DMPK | 3500.0 | nM |
| Ruxolitinib | DRAK2 | 3500.0 | nM |