INCB018424 KINOMEscan - Dataset (ID:20173)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | KIT | nM | |
Ruxolitinib | KIT(A829P) | 6300.0 | nM |
Ruxolitinib | KIT(D816H) | 6300.0 | nM |
Ruxolitinib | KIT(D816V) | 7100.0 | nM |
Ruxolitinib | KIT(L576P) | nM | |
Ruxolitinib | KIT(V559D) | nM | |
Ruxolitinib | KIT(V559D,T670I) | nM | |
Ruxolitinib | KIT(V559D,V654A) | nM | |
Ruxolitinib | LATS1 | nM | |
Ruxolitinib | LATS2 | nM | |
Ruxolitinib | LCK | nM | |
Ruxolitinib | LIMK1 | nM | |
Ruxolitinib | LIMK2 | nM | |
Ruxolitinib | LKB1 | nM | |
Ruxolitinib | LOK | nM | |
Ruxolitinib | LRRK2 | 290.0 | nM |
Ruxolitinib | LRRK2(G2019S) | 90.0 | nM |
Ruxolitinib | LTK | 440.0 | nM |
Ruxolitinib | LYN | nM | |
Ruxolitinib | M3K13 | nM | |
Ruxolitinib | MAK | nM | |
Ruxolitinib | MAP3K1 | 4200.0 | nM |
Ruxolitinib | MAP3K15 | 1100.0 | nM |
Ruxolitinib | M3K2 | 41.0 | nM |
Ruxolitinib | MAP3K3 | 150.0 | nM |