INCB018424 KINOMEscan - Dataset (ID:20173)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | HCK | nM | |
Ruxolitinib | HIPK1 | 1200.0 | nM |
Ruxolitinib | HIPK2 | 1000.0 | nM |
Ruxolitinib | HIPK3 | 1200.0 | nM |
Ruxolitinib | HIPK4 | nM | |
Ruxolitinib | M4K1 | nM | |
Ruxolitinib | HUNK | nM | |
Ruxolitinib | ICK | nM | |
Ruxolitinib | IGF1R | nM | |
Ruxolitinib | IKKA | nM | |
Ruxolitinib | IKKB | 2300.0 | nM |
Ruxolitinib | IKKE | 1200.0 | nM |
Ruxolitinib | INSR | nM | |
Ruxolitinib | INSRR | nM | |
Ruxolitinib | IRAK1 | 290.0 | nM |
Ruxolitinib | IRAK3 | nM | |
Ruxolitinib | IRAK4 | nM | |
Ruxolitinib | ITK | nM | |
Ruxolitinib | JAK1(JH1domain-catalytic) | 3.4 | nM |
Ruxolitinib | JAK1(JH2domain-pseudokinase) | nM | |
Ruxolitinib | JAK2(JH1domain-catalytic) | 0.0 | nM |
Ruxolitinib | JAK3(JH1domain-catalytic) | 2.0 | nM |
Ruxolitinib | JNK1 | 4800.0 | nM |
Ruxolitinib | MK09 | nM | |
Ruxolitinib | JNK3 | nM |