BIBW-2992 KINOMEscan - Dataset (ID:20172)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Afatinib | DCAMKL2 | nM | |
| Afatinib | DCAMKL3 | nM | |
| Afatinib | DDR1 | nM | |
| Afatinib | DDR2 | nM | |
| Afatinib | M3K12 | nM | |
| Afatinib | DMPK | nM | |
| Afatinib | DMPK2 | nM | |
| Afatinib | DRAK1 | 2300.0 | nM |
| Afatinib | DRAK2 | nM | |
| Afatinib | DYRK1A | 970.0 | nM |
| Afatinib | DYRK1B | 2800.0 | nM |
| Afatinib | DYRK2 | 1800.0 | nM |
| Afatinib | EGFR | 0.3 | nM |
| Afatinib | EGFR(E746-A750del) | 0.1 | nM |
| Afatinib | EGFR(G719C) | 0.1 | nM |
| Afatinib | EGFR(G719S) | 0.2 | nM |
| Afatinib | EGFR(L747-E749del, A750P) | 0.1 | nM |
| Afatinib | EGFR(L747-S752del, P753S) | 0.1 | nM |
| Afatinib | EGFR(L747-T751del,Sins) | 0.1 | nM |
| Afatinib | EGFR(L858R) | 0.2 | nM |
| Afatinib | EGFR(L858R,T790M) | 1.1 | nM |
| Afatinib | EGFR(L861Q) | 0.2 | nM |
| Afatinib | EGFR(S752-I759del) | 0.1 | nM |
| Afatinib | EGFR(T790M) | 0.6 | nM |
| Afatinib | EIF2AK1 | nM |