BIBW-2992 KINOMEscan - Dataset (ID:20172)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Afatinib | AAK1 | nM | |
| Afatinib | ABL1(E255K)-phosphorylated | 420.0 | nM |
| Afatinib | ABL1(F317I)-nonphosphorylated | 2900.0 | nM |
| Afatinib | ABL1(F317I)-phosphorylated | 750.0 | nM |
| Afatinib | ABL1(F317L)-nonphosphorylated | 580.0 | nM |
| Afatinib | ABL1(F317L)-phosphorylated | 230.0 | nM |
| Afatinib | ABL1(H396P)-nonphosphorylated | 500.0 | nM |
| Afatinib | ABL1(H396P)-phosphorylated | 500.0 | nM |
| Afatinib | ABL1(M351T)-phosphorylated | 1200.0 | nM |
| Afatinib | ABL1(Q252H)-nonphosphorylated | 790.0 | nM |
| Afatinib | ABL1(Q252H)-phosphorylated | 380.0 | nM |
| Afatinib | ABL1(T315I)-nonphosphorylated | 2600.0 | nM |
| Afatinib | ABL1(T315I)-phosphorylated | 870.0 | nM |
| Afatinib | ABL1(Y253F)-phosphorylated | 830.0 | nM |
| Afatinib | ABL1-nonphosphorylated | 1300.0 | nM |
| Afatinib | ABL1-phosphorylated | 570.0 | nM |
| Afatinib | ABL2 | nM | |
| Afatinib | ACVR1 | nM | |
| Afatinib | ACVR1B | nM | |
| Afatinib | ACVR2A | nM | |
| Afatinib | ACVR2B | nM | |
| Afatinib | ACVRL1 | nM | |
| Afatinib | ADCK3 | nM | |
| Afatinib | ADCK4 | nM | |
| Afatinib | AKT1 | nM |