BIBW-2992 KINOMEscan - Dataset (ID:20172)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Afatinib | PRKX | nM | |
Afatinib | PRP4 | nM | |
Afatinib | FAK2 | nM | |
Afatinib | SIK3 | nM | |
Afatinib | RAF1 | nM | |
Afatinib | RET | nM | |
Afatinib | RET(M918T) | nM | |
Afatinib | RET(V804L) | nM | |
Afatinib | RET(V804M) | nM | |
Afatinib | RIOK1 | nM | |
Afatinib | RIOK2 | nM | |
Afatinib | RIOK3 | nM | |
Afatinib | RIPK1 | nM | |
Afatinib | RIPK2 | 2700.0 | nM |
Afatinib | RIPK4 | nM | |
Afatinib | RIPK5 | nM | |
Afatinib | ROCK1 | nM | |
Afatinib | ROCK2 | nM | |
Afatinib | ROS1 | nM | |
Afatinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
Afatinib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
Afatinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
Afatinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Afatinib | RSK1(Kin.Dom.1-N-terminal) | nM | |
Afatinib | RSK1(Kin.Dom.2-C-terminal) | nM |