BIBW-2992 KINOMEscan - Dataset (ID:20172)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Afatinib | FLT3(N841I) | 6200.0 | nM |
| Afatinib | MET(M1250T) | 6000.0 | nM |
| Afatinib | AXL | 5300.0 | nM |
| Afatinib | SBK1 | 4800.0 | nM |
| Afatinib | ERBB3 | 4500.0 | nM |
| Afatinib | LOK | 4300.0 | nM |
| Afatinib | SLK | 3700.0 | nM |
| Afatinib | EPHB6 | 3100.0 | nM |
| Afatinib | TXK | 3100.0 | nM |
| Afatinib | RSK4(Kin.Dom.2-C-terminal) | 3100.0 | nM |
| Afatinib | ABL1(F317I)-nonphosphorylated | 2900.0 | nM |
| Afatinib | CIT | 2900.0 | nM |
| Afatinib | DYRK1B | 2800.0 | nM |
| Afatinib | SRC | 2800.0 | nM |
| Afatinib | RIPK2 | 2700.0 | nM |
| Afatinib | MET(Y1235D) | 2600.0 | nM |
| Afatinib | ABL1(T315I)-nonphosphorylated | 2600.0 | nM |
| Afatinib | DRAK1 | 2300.0 | nM |
| Afatinib | HCK | 2200.0 | nM |
| Afatinib | MET | 2200.0 | nM |
| Afatinib | MK09 | 2100.0 | nM |
| Afatinib | JNK3 | 2000.0 | nM |
| Afatinib | DYRK2 | 1800.0 | nM |
| Afatinib | FLT3(D835H) | 1800.0 | nM |
| Afatinib | MKNK1 | 1800.0 | nM |