BIBW-2992 KINOMEscan - Dataset (ID:20172)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Afatinib | EGFR(L747-T751del,Sins) | 0.1 | nM |
Afatinib | EGFR(S752-I759del) | 0.1 | nM |
Afatinib | EGFR(G719C) | 0.1 | nM |
Afatinib | EGFR(L747-E749del, A750P) | 0.1 | nM |
Afatinib | EGFR(L747-S752del, P753S) | 0.1 | nM |
Afatinib | EGFR(E746-A750del) | 0.1 | nM |
Afatinib | EGFR(L861Q) | 0.2 | nM |
Afatinib | EGFR(G719S) | 0.2 | nM |
Afatinib | EGFR(L858R) | 0.2 | nM |
Afatinib | EGFR | 0.3 | nM |
Afatinib | EGFR(T790M) | 0.6 | nM |
Afatinib | EGFR(L858R,T790M) | 1.1 | nM |
Afatinib | ERBB2 | 5.0 | nM |
Afatinib | ERBB4 | 6.3 | nM |
Afatinib | GAK | 79.0 | nM |
Afatinib | BLK | 220.0 | nM |
Afatinib | ABL1(F317L)-phosphorylated | 230.0 | nM |
Afatinib | IRAK1 | 240.0 | nM |
Afatinib | EPHA6 | 340.0 | nM |
Afatinib | HIPK4 | 360.0 | nM |
Afatinib | ABL1(Q252H)-phosphorylated | 380.0 | nM |
Afatinib | ABL1(E255K)-phosphorylated | 420.0 | nM |
Afatinib | PHKG2 | 470.0 | nM |
Afatinib | ABL1(H396P)-nonphosphorylated | 500.0 | nM |
Afatinib | ABL1(H396P)-phosphorylated | 500.0 | nM |