AB-1010 KINOMEscan - Dataset (ID:20170)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Masitinib | EGFR(L861Q) | 4700.0 | nM |
| Masitinib | EPHA3 | 2500.0 | nM |
| Masitinib | BRAF(V600E) | 1800.0 | nM |
| Masitinib | EPHA8 | 1800.0 | nM |
| Masitinib | RIOK2 | 1700.0 | nM |
| Masitinib | KIT(D816H) | 1500.0 | nM |
| Masitinib | PIM1 | 1300.0 | nM |
| Masitinib | EGFR(L747-T751del,Sins) | 1300.0 | nM |
| Masitinib | KIT(D816V) | 1300.0 | nM |
| Masitinib | ERBB2 | 1200.0 | nM |
| Masitinib | SRC | 900.0 | nM |
| Masitinib | EGFR(L747-E749del, A750P) | 800.0 | nM |
| Masitinib | MLTK | 770.0 | nM |
| Masitinib | PIM3 | 720.0 | nM |
| Masitinib | HCK | 690.0 | nM |
| Masitinib | FGR | 640.0 | nM |
| Masitinib | YES | 570.0 | nM |
| Masitinib | BLK | 150.0 | nM |
| Masitinib | FYN | 140.0 | nM |
| Masitinib | ABL1(M351T)-phosphorylated | 140.0 | nM |
| Masitinib | ABL1(E255K)-phosphorylated | 140.0 | nM |
| Masitinib | ABL1(H396P)-phosphorylated | 140.0 | nM |
| Masitinib | ABL1(F317L)-phosphorylated | 110.0 | nM |
| Masitinib | ABL2 | 110.0 | nM |
| Masitinib | FRK | 87.0 | nM |