AB-1010 KINOMEscan - Dataset (ID:20170)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Masitinib | ABL1-nonphosphorylated | 2.1 | nM |
Masitinib | ABL1(Q252H)-phosphorylated | 4.6 | nM |
Masitinib | KIT(V559D,V654A) | 4.7 | nM |
Masitinib | KIT(V559D) | 5.8 | nM |
Masitinib | ABL1(Q252H)-nonphosphorylated | 6.0 | nM |
Masitinib | CSF1R | 7.6 | nM |
Masitinib | KIT(L576P) | 7.9 | nM |
Masitinib | ABL1(F317I)-nonphosphorylated | 8.0 | nM |
Masitinib | KIT | 8.1 | nM |
Masitinib | PGFRB | 8.4 | nM |
Masitinib | DDR1 | 8.7 | nM |
Masitinib | ABL1(F317L)-nonphosphorylated | 10.0 | nM |
Masitinib | ABL1(H396P)-nonphosphorylated | 11.0 | nM |
Masitinib | KIT(A829P) | 12.0 | nM |
Masitinib | ABL1(Y253F)-phosphorylated | 25.0 | nM |
Masitinib | PGFRA | 25.0 | nM |
Masitinib | DDR2 | 26.0 | nM |
Masitinib | LCK | 31.0 | nM |
Masitinib | ABL1-phosphorylated | 55.0 | nM |
Masitinib | LYN | 61.0 | nM |
Masitinib | ABL1(F317I)-phosphorylated | 78.0 | nM |
Masitinib | FRK | 87.0 | nM |
Masitinib | ABL1(F317L)-phosphorylated | 110.0 | nM |
Masitinib | ABL2 | 110.0 | nM |
Masitinib | FYN | 140.0 | nM |