AB-1010 KINOMEscan - Dataset (ID:20170)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Masitinib | AAK1 | nM | |
| Masitinib | ABL1(E255K)-phosphorylated | 140.0 | nM |
| Masitinib | ABL1(F317I)-nonphosphorylated | 8.0 | nM |
| Masitinib | ABL1(F317I)-phosphorylated | 78.0 | nM |
| Masitinib | ABL1(F317L)-nonphosphorylated | 10.0 | nM |
| Masitinib | ABL1(F317L)-phosphorylated | 110.0 | nM |
| Masitinib | ABL1(H396P)-nonphosphorylated | 11.0 | nM |
| Masitinib | ABL1(H396P)-phosphorylated | 140.0 | nM |
| Masitinib | ABL1(M351T)-phosphorylated | 140.0 | nM |
| Masitinib | ABL1(Q252H)-nonphosphorylated | 6.0 | nM |
| Masitinib | ABL1(Q252H)-phosphorylated | 4.6 | nM |
| Masitinib | ABL1(T315I)-nonphosphorylated | nM | |
| Masitinib | ABL1(T315I)-phosphorylated | nM | |
| Masitinib | ABL1(Y253F)-phosphorylated | 25.0 | nM |
| Masitinib | ABL1-nonphosphorylated | 2.1 | nM |
| Masitinib | ABL1-phosphorylated | 55.0 | nM |
| Masitinib | ABL2 | 110.0 | nM |
| Masitinib | ACVR1 | nM | |
| Masitinib | ACVR1B | nM | |
| Masitinib | ACVR2A | nM | |
| Masitinib | ACVR2B | nM | |
| Masitinib | ACVRL1 | nM | |
| Masitinib | ADCK3 | nM | |
| Masitinib | ADCK4 | nM | |
| Masitinib | AKT1 | nM |