CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Canertinib | DCAMKL2 | nM | |
| Canertinib | DCAMKL3 | nM | |
| Canertinib | DDR1 | 400.00 | nM |
| Canertinib | DDR2 | nM | |
| Canertinib | M3K12 | nM | |
| Canertinib | DMPK | 7000.00 | nM |
| Canertinib | DMPK2 | nM | |
| Canertinib | DRAK1 | nM | |
| Canertinib | DRAK2 | 7300.00 | nM |
| Canertinib | DYRK1A | 1500.00 | nM |
| Canertinib | DYRK1B | nM | |
| Canertinib | DYRK2 | 6700.00 | nM |
| Canertinib | EGFR | 0.19 | nM |
| Canertinib | EGFR(E746-A750del) | 0.26 | nM |
| Canertinib | EGFR(G719C) | 0.13 | nM |
| Canertinib | EGFR(G719S) | 0.19 | nM |
| Canertinib | EGFR(L747-E749del, A750P) | 0.17 | nM |
| Canertinib | EGFR(L747-S752del, P753S) | 0.26 | nM |
| Canertinib | EGFR(L747-T751del,Sins) | 0.26 | nM |
| Canertinib | EGFR(L858R) | 0.24 | nM |
| Canertinib | EGFR(L858R,T790M) | 0.28 | nM |
| Canertinib | EGFR(L861Q) | 0.22 | nM |
| Canertinib | EGFR(S752-I759del) | 0.19 | nM |
| Canertinib | EGFR(T790M) | 0.10 | nM |
| Canertinib | EIF2AK1 | nM |