CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Canertinib | PRKX | nM | |
Canertinib | PRP4 | nM | |
Canertinib | FAK2 | nM | |
Canertinib | SIK3 | 700.00 | nM |
Canertinib | RAF1 | nM | |
Canertinib | RET | 4200.00 | nM |
Canertinib | RET(M918T) | 840.00 | nM |
Canertinib | RET(V804L) | nM | |
Canertinib | RET(V804M) | nM | |
Canertinib | RIOK1 | 8400.00 | nM |
Canertinib | RIOK2 | nM | |
Canertinib | RIOK3 | nM | |
Canertinib | RIPK1 | nM | |
Canertinib | RIPK2 | 300.00 | nM |
Canertinib | RIPK4 | nM | |
Canertinib | RIPK5 | nM | |
Canertinib | ROCK1 | nM | |
Canertinib | ROCK2 | nM | |
Canertinib | ROS1 | nM | |
Canertinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
Canertinib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
Canertinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
Canertinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Canertinib | RSK1(Kin.Dom.1-N-terminal) | nM | |
Canertinib | RSK1(Kin.Dom.2-C-terminal) | 6200.00 | nM |