CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Canertinib | AAK1 | nM | |
| Canertinib | ABL1(E255K)-phosphorylated | 30.00 | nM |
| Canertinib | ABL1(F317I)-nonphosphorylated | 3200.00 | nM |
| Canertinib | ABL1(F317I)-phosphorylated | 1000.00 | nM |
| Canertinib | ABL1(F317L)-nonphosphorylated | 1500.00 | nM |
| Canertinib | ABL1(F317L)-phosphorylated | 91.00 | nM |
| Canertinib | ABL1(H396P)-nonphosphorylated | 46.00 | nM |
| Canertinib | ABL1(H396P)-phosphorylated | 57.00 | nM |
| Canertinib | ABL1(M351T)-phosphorylated | 38.00 | nM |
| Canertinib | ABL1(Q252H)-nonphosphorylated | 91.00 | nM |
| Canertinib | ABL1(Q252H)-phosphorylated | 22.00 | nM |
| Canertinib | ABL1(T315I)-nonphosphorylated | 690.00 | nM |
| Canertinib | ABL1(T315I)-phosphorylated | 69.00 | nM |
| Canertinib | ABL1(Y253F)-phosphorylated | 42.00 | nM |
| Canertinib | ABL1-nonphosphorylated | 210.00 | nM |
| Canertinib | ABL1-phosphorylated | 30.00 | nM |
| Canertinib | ABL2 | 870.00 | nM |
| Canertinib | ACVR1 | 1700.00 | nM |
| Canertinib | ACVR1B | nM | |
| Canertinib | ACVR2A | nM | |
| Canertinib | ACVR2B | nM | |
| Canertinib | ACVRL1 | nM | |
| Canertinib | ADCK3 | 1500.00 | nM |
| Canertinib | ADCK4 | 3400.00 | nM |
| Canertinib | AKT1 | nM |