Gefitinib KINOMEscan - Dataset (ID:20161)

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Small Molecule Protein Kd Conc unit
Gefitinib EPHA1 4000.0
nM
Gefitinib EPHA2
nM
Gefitinib EPHA3 5500.0
nM
Gefitinib EPHA4
nM
Gefitinib EPHA5 1500.0
nM
Gefitinib EPHA6 590.0
nM
Gefitinib EPHA7
nM
Gefitinib EPHA8 1800.0
nM
Gefitinib EPHB1 1300.0
nM
Gefitinib EPHB2
nM
Gefitinib EPHB3
nM
Gefitinib EPHB4 2500.0
nM
Gefitinib EPHB6 3200.0
nM
Gefitinib ERBB2 3500.0
nM
Gefitinib ERBB3 790.0
nM
Gefitinib ERBB4 410.0
nM
Gefitinib MK03
nM
Gefitinib MK01
nM
Gefitinib ERK3 1600.0
nM
Gefitinib ERK4 3100.0
nM
Gefitinib ERK5
nM
Gefitinib ERK8
nM
Gefitinib ERN1
nM
Gefitinib FAK1
nM
Gefitinib FER
nM