Gefitinib KINOMEscan - Dataset (ID:20161)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Gefitinib | DCAMKL2 | nM | |
| Gefitinib | DCAMKL3 | 2900.0 | nM |
| Gefitinib | DDR1 | nM | |
| Gefitinib | DDR2 | nM | |
| Gefitinib | M3K12 | nM | |
| Gefitinib | DMPK | 6900.0 | nM |
| Gefitinib | DMPK2 | nM | |
| Gefitinib | DRAK1 | 2000.0 | nM |
| Gefitinib | DRAK2 | 3800.0 | nM |
| Gefitinib | DYRK1A | nM | |
| Gefitinib | DYRK1B | nM | |
| Gefitinib | DYRK2 | nM | |
| Gefitinib | EGFR | 1.0 | nM |
| Gefitinib | EGFR(E746-A750del) | 0.5 | nM |
| Gefitinib | EGFR(G719C) | 2.0 | nM |
| Gefitinib | EGFR(G719S) | 1.1 | nM |
| Gefitinib | EGFR(L747-E749del, A750P) | 0.6 | nM |
| Gefitinib | EGFR(L747-S752del, P753S) | 0.6 | nM |
| Gefitinib | EGFR(L747-T751del,Sins) | 0.5 | nM |
| Gefitinib | EGFR(L858R) | 0.9 | nM |
| Gefitinib | EGFR(L858R,T790M) | 140.0 | nM |
| Gefitinib | EGFR(L861Q) | 1.4 | nM |
| Gefitinib | EGFR(S752-I759del) | 1.0 | nM |
| Gefitinib | EGFR(T790M) | 40.0 | nM |
| Gefitinib | EIF2AK1 | nM |