Gefitinib KINOMEscan - Dataset (ID:20161)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Gefitinib | PRKX | nM | |
Gefitinib | PRP4 | nM | |
Gefitinib | FAK2 | nM | |
Gefitinib | SIK3 | nM | |
Gefitinib | RAF1 | nM | |
Gefitinib | RET | nM | |
Gefitinib | RET(M918T) | nM | |
Gefitinib | RET(V804L) | nM | |
Gefitinib | RET(V804M) | nM | |
Gefitinib | RIOK1 | nM | |
Gefitinib | RIOK2 | nM | |
Gefitinib | RIOK3 | nM | |
Gefitinib | RIPK1 | nM | |
Gefitinib | RIPK2 | 530.0 | nM |
Gefitinib | RIPK4 | nM | |
Gefitinib | RIPK5 | nM | |
Gefitinib | ROCK1 | nM | |
Gefitinib | ROCK2 | nM | |
Gefitinib | ROS1 | nM | |
Gefitinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
Gefitinib | RPS6KA4(Kin.Dom.2-C-terminal) | 1200.0 | nM |
Gefitinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
Gefitinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Gefitinib | RSK1(Kin.Dom.1-N-terminal) | nM | |
Gefitinib | RSK1(Kin.Dom.2-C-terminal) | nM |