Gefitinib KINOMEscan - Dataset (ID:20161)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Gefitinib | FES | nM | |
Gefitinib | FGFR1 | nM | |
Gefitinib | FGFR2 | nM | |
Gefitinib | FGFR3 | nM | |
Gefitinib | FGFR3(G697C) | nM | |
Gefitinib | FGFR4 | nM | |
Gefitinib | FGR | 2600.0 | nM |
Gefitinib | VGFR1 | nM | |
Gefitinib | FLT3 | 3100.0 | nM |
Gefitinib | FLT3(D835H) | 1100.0 | nM |
Gefitinib | FLT3(D835Y) | 1000.0 | nM |
Gefitinib | FLT3(ITD) | 2900.0 | nM |
Gefitinib | FLT3(K663Q) | 5100.0 | nM |
Gefitinib | FLT3(N841I) | 3000.0 | nM |
Gefitinib | FLT3(R834Q) | 3500.0 | nM |
Gefitinib | FLT4 | nM | |
Gefitinib | FRK | 2000.0 | nM |
Gefitinib | FYN | nM | |
Gefitinib | GAK | 13.0 | nM |
Gefitinib | GCN2(Kin.Dom.2,S808G) | nM | |
Gefitinib | GRK1 | nM | |
Gefitinib | GRK4 | nM | |
Gefitinib | GRK7 | nM | |
Gefitinib | GSK3A | nM | |
Gefitinib | GSK3B | nM |