Gefitinib KINOMEscan - Dataset (ID:20161)

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Small Molecule Protein Kd Conc unit
Gefitinib FES
nM
Gefitinib FGFR1
nM
Gefitinib FGFR2
nM
Gefitinib FGFR3
nM
Gefitinib FGFR3(G697C)
nM
Gefitinib FGFR4
nM
Gefitinib FGR 2600.0
nM
Gefitinib VGFR1
nM
Gefitinib FLT3 3100.0
nM
Gefitinib FLT3(D835H) 1100.0
nM
Gefitinib FLT3(D835Y) 1000.0
nM
Gefitinib FLT3(ITD) 2900.0
nM
Gefitinib FLT3(K663Q) 5100.0
nM
Gefitinib FLT3(N841I) 3000.0
nM
Gefitinib FLT3(R834Q) 3500.0
nM
Gefitinib FLT4
nM
Gefitinib FRK 2000.0
nM
Gefitinib FYN
nM
Gefitinib GAK 13.0
nM
Gefitinib GCN2(Kin.Dom.2,S808G)
nM
Gefitinib GRK1
nM
Gefitinib GRK4
nM
Gefitinib GRK7
nM
Gefitinib GSK3A
nM
Gefitinib GSK3B
nM