NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NPK76-II-72-1 | PC-3 | MAP2K6 | DVkPSNVLINALGQVK | Lys2 | -8.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | MAP2K6 | HVPSGQIMAVkR | Lys1 | 2.5 | 10 | uM |
NPK76-II-72-1 | HeLa | MAP3K1 | DVkGANLLIDSTGQR | Lys2 | -6.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -82.4 | 10 | uM |
NPK76-II-72-1 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | -18.8 | 10 | uM |
NPK76-II-72-1 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 3.8 | 10 | uM |
NPK76-II-72-1 | HeLa | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -16.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 3.7 | 10 | uM |
NPK76-II-72-1 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | -11.7 | 10 | uM |
NPK76-II-72-1 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | -44.8 | 10 | uM |
NPK76-II-72-1 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 1.4 | 10 | uM |
NPK76-II-72-1 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 5.7 | 10 | uM |
NPK76-II-72-1 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | -7.8 | 10 | uM |
NPK76-II-72-1 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | -3.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 6.5 | 10 | uM |
NPK76-II-72-1 | HeLa | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | -21.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | -11.5 | 10 | uM |
NPK76-II-72-1 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -9.4 | 10 | uM |
NPK76-II-72-1 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -0.9 | 10 | uM |
NPK76-II-72-1 | HeLa | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | -5.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | -12.6 | 10 | uM |
NPK76-II-72-1 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | -9.4 | 10 | uM |
NPK76-II-72-1 | HeLa | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | -18.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 4.9 | 10 | uM |
NPK76-II-72-1 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | -8.3 | 10 | uM |