NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NPK76-II-72-1 PC-3 MAP2K6
DVkPSNVLINALGQVK
Lys2
-8.0
10
uM
NPK76-II-72-1 PC-3 MAP2K6
HVPSGQIMAVkR
Lys1
2.5
10
uM
NPK76-II-72-1 HeLa MAP3K1
DVkGANLLIDSTGQR
Lys2
-6.5
10
uM
NPK76-II-72-1 PC-3 M3K2
ELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-82.4
10
uM
NPK76-II-72-1 HeLa M3K2,MAP3K3
DIkGANILR
Lys2
-18.8
10
uM
NPK76-II-72-1 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
3.8
10
uM
NPK76-II-72-1 HeLa MAP3K4
DIkGANIFLTSSGLIK
Lys2
-16.2
10
uM
NPK76-II-72-1 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
3.7
10
uM
NPK76-II-72-1 HeLa MAP3K5,MAP3K6,MAP3K7
IAIkEIPERDSR
Lys1
-11.7
10
uM
NPK76-II-72-1 HeLa MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
-44.8
10
uM
NPK76-II-72-1 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
1.4
10
uM
NPK76-II-72-1 HeLa MAST3
DLkPDNLLITSLGHIK
Lys2
5.7
10
uM
NPK76-II-72-1 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
-7.8
10
uM
NPK76-II-72-1 HeLa MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
-3.5
10
uM
NPK76-II-72-1 PC-3 MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
6.5
10
uM
NPK76-II-72-1 HeLa MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
-21.3
10
uM
NPK76-II-72-1 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
-11.5
10
uM
NPK76-II-72-1 HeLa MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
-9.4
10
uM
NPK76-II-72-1 HeLa MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
-0.9
10
uM
NPK76-II-72-1 HeLa MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
-5.3
10
uM
NPK76-II-72-1 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
-12.6
10
uM
NPK76-II-72-1 PC-3 MST1,MST2
DIkAGNILLNTEGHAK
Lys2
-9.4
10
uM
NPK76-II-72-1 HeLa MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
-18.5
10
uM
NPK76-II-72-1 PC-3 MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
4.9
10
uM
NPK76-II-72-1 HeLa MST3
DIkAANVLLSEHGEVK
Lys2
-8.3
10
uM