NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -31.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | -1.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -1.8 | 10 | uM |
| NPK76-II-72-1 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -14.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | -30.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 20.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -2.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | ATR | FYIMMCkPK | ATP | -80.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | ATR | FYIMMCkPK | ATP | 7.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -6.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 10.8 | 10 | uM |
| NPK76-II-72-1 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 63.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 64.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | -33.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | -14.6 | 10 | uM |
| NPK76-II-72-1 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 0.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -10.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | 3.6 | 10 | uM |
| NPK76-II-72-1 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -6.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | -9.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CHK2 | VAIkIISK | Lys1 | 31.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -2.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | 14.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -5.2 | 10 | uM |