NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -5.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -5.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 16.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | -4.7 | 10 | uM |
| NPK76-II-72-1 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | -28.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | -2.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -0.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -58.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | 10.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | -13.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | 3.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MK11 | QELNkTVWEVPQR | Other | -46.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PDK1 | EYAIkILEK | Lys1 | 22.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 31.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | PKD2 | DVAVkVIDK | Lys1 | -11.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | RIPK3 | DLkPSNVLLDPELHVK | Lys2 | -1.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | -26.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | -11.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | SLK | ETSVLAAAkVIDTK | Lys1 | 68.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | SYK | ISDFGLSkALR | Activation Loop | -12.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | -9.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -2.6 | 10 | uM |