NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NPK76-II-72-1 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | -6.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | -0.5 | 10 | uM |
NPK76-II-72-1 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -0.3 | 10 | uM |
NPK76-II-72-1 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -8.7 | 10 | uM |
NPK76-II-72-1 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -7.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | -4.5 | 10 | uM |
NPK76-II-72-1 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -6.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | -7.8 | 10 | uM |
NPK76-II-72-1 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -20.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 10.3 | 10 | uM |
NPK76-II-72-1 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -4.8 | 10 | uM |
NPK76-II-72-1 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -17.9 | 10 | uM |
NPK76-II-72-1 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -19.9 | 10 | uM |
NPK76-II-72-1 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -10.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -6.5 | 10 | uM |
NPK76-II-72-1 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -10.1 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -9.4 | 10 | uM |
NPK76-II-72-1 | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -5.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK14 | LVALkVIR | Lys1 | 3.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 6.1 | 10 | uM |
NPK76-II-72-1 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 0.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 0.6 | 10 | uM |
NPK76-II-72-1 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -7.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -0.3 | 10 | uM |