NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NPK76-II-72-1 PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
-6.0
10
uM
NPK76-II-72-1 PC-3 NDR2
DTGHIYAMkILR
Lys1
-0.5
10
uM
NPK76-II-72-1 HeLa NEK1
DIkSQNIFLTK
Lys2
-0.3
10
uM
NPK76-II-72-1 HeLa NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-8.7
10
uM
NPK76-II-72-1 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-7.4
10
uM
NPK76-II-72-1 PC-3 NEK8
DLkTQNILLDK
Lys2
-4.5
10
uM
NPK76-II-72-1 HeLa NEK9
DIkTLNIFLTK
Lys2
-6.5
10
uM
NPK76-II-72-1 PC-3 NEK9
DIkTLNIFLTK
Lys2
-7.8
10
uM
NPK76-II-72-1 HeLa NEK9
LGDYGLAkK
Activation Loop
-20.0
10
uM
NPK76-II-72-1 PC-3 NEK9
LGDYGLAkK
Activation Loop
10.3
10
uM
NPK76-II-72-1 HeLa p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-4.8
10
uM
NPK76-II-72-1 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-17.9
10
uM
NPK76-II-72-1 HeLa KS6B1
DLkPENIMLNHQGHVK
Lys2
-19.9
10
uM
NPK76-II-72-1 PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
-10.2
10
uM
NPK76-II-72-1 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-6.5
10
uM
NPK76-II-72-1 HeLa KS6B2
DLkPENIMLSSQGHIK
Lys2
-10.1
10
uM
NPK76-II-72-1 PC-3 CDK16
LTDNLVALkEIR
Lys1
-9.4
10
uM
NPK76-II-72-1 HeLa PCTAIRE2
DLkPQNLLINEK
Lys2
-5.0
10
uM
NPK76-II-72-1 PC-3 CDK14
LVALkVIR
Lys1
3.0
10
uM
NPK76-II-72-1 PC-3 PHKg2
ATGHEFAVkIMEVTAER
Lys1
6.1
10
uM
NPK76-II-72-1 HeLa PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
0.2
10
uM
NPK76-II-72-1 PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
0.6
10
uM
NPK76-II-72-1 HeLa PI4KB
VPHTQAVVLNSkDK
ATP
-7.0
10
uM
NPK76-II-72-1 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
0.4
10
uM
NPK76-II-72-1 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-0.3
10
uM