NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | PC-3 | ILK | WQGNDIVVkVLK | Lys1 | -18.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | IRAK1 | AIQFLHQDSPSLIHGDIkSSNVLLDER | Lys2 | -6.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -7.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -8.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -3.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 84.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -12.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -25.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -11.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -7.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | 0.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | LATS1 | ALYATkTLR | Lys1 | -22.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -14.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 7.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | -0.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | LOK | NKETGALAAAkVIETK | Lys1 | 46.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | LOK | NKETGALAAAkVIETK | Lys1 | 34.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -17.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | 4.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | -16.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MAP2K3 | DVkPSNVLINK | Lys2 | -12.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MAP2K4 | MVHKPSGQIMAVkR | Lys1 | -8.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | -11.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | MAP2K6 | DVkPSNVLINALGQVK | Lys2 | -47.1 | 10 | uM |