NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

 Full screen view
Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
3.3
 0.05
uM
NVP-BHG712 PC-3 MLK4
DLkSSNILLLEK
Lys2
-1.7
 0.05
uM
NVP-BHG712 PC-3 MLKL
APVAIkVFK
Lys1
14.7
 0.05
uM
NVP-BHG712 PC-3 MRCKb
DIkPDNVLLDVNGHIR
Lys2
17.6
 0.05
uM
NVP-BHG712 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
-26.4
 0.05
uM
NVP-BHG712 PC-3 MSK1 domain1
LGIIYRDIkLENILLDSNGHVVLTDFGLSK
Lys2
-14.2
 0.05
uM
NVP-BHG712 PC-3 MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
-0.8
 0.05
uM
NVP-BHG712 PC-3 MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
-5.6
 0.05
uM
NVP-BHG712 PC-3 MSK2 domain1
DLkLENVLLDSEGHIVLTDFGLSK
Lys2
-3.1
 0.05
uM
NVP-BHG712 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
6.8
 0.05
uM
NVP-BHG712 PC-3 MST1,MST2
DIkAGNILLNTEGHAK
Lys2
5.6
 0.05
uM
NVP-BHG712 PC-3 MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
6.8
 0.05
uM
NVP-BHG712 PC-3 MST3
DIkAANVLLSEHGEVK
Lys2
0.7
 0.05
uM
NVP-BHG712 PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
-1.1
 0.05
uM
NVP-BHG712 PC-3 NDR1
DTGHVYAMkILR
Lys1
-8.5
 0.05
uM
NVP-BHG712 PC-3 NDR2
DTGHIYAMkILR
Lys1
2.6
 0.05
uM
NVP-BHG712 PC-3 NDR2
DIkPDNLLLDAK
Lys2
-3.0
 0.05
uM
NVP-BHG712 PC-3 NEK1
DIkSQNIFLTK
Lys2
-4.2
 0.05
uM
NVP-BHG712 PC-3 NEK4
DLkTQNVFLTR
Lys2
0.4
 0.05
uM
NVP-BHG712 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
10.7
 0.05
uM
NVP-BHG712 PC-3 NEK7
AACLLDGVPVALkK
Lys1
4.0
 0.05
uM
NVP-BHG712 PC-3 NEK8
DLkTQNILLDK
Lys2
-8.2
 0.05
uM
NVP-BHG712 PC-3 NEK9
LGDYGLAkK
Activation Loop
1.5
 0.05
uM
NVP-BHG712 PC-3 NEK9
TEDDSLVVWkEVDLTR
Lys1
-0.3
 0.05
uM
NVP-BHG712 PC-3 NEK9
DIkTLNIFLTK
Lys2
-11.3
 0.05
uM