NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
2.6
 0.05
uM
NVP-BHG712 PC-3 MAP2K3
MCDFGISGYLVDSVAkTMDAGCKPYMAPER
Activation Loop
-4.8
 0.05
uM
NVP-BHG712 PC-3 MAP2K3
DVkPSNVLINK
Lys2
5.5
 0.05
uM
NVP-BHG712 PC-3 MAP2K4
LCDFGISGQLVDSIAkTR
Activation Loop
-9.4
 0.05
uM
NVP-BHG712 PC-3 MAP2K4
DIkPSNILLDR
Lys2
17.0
 0.05
uM
NVP-BHG712 PC-3 MAP2K5
DVkPSNMLVNTR
Lys2
-14.1
 0.05
uM
NVP-BHG712 PC-3 MAP2K6
HVPSGQIMAVkR
Lys1
-13.3
 0.05
uM
NVP-BHG712 PC-3 MAP2K6
DVkPSNVLINALGQVK
Lys2
4.9
 0.05
uM
NVP-BHG712 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-18.8
 0.05
uM
NVP-BHG712 PC-3 M3K2
ELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
2.8
 0.05
uM
NVP-BHG712 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
-12.5
 0.05
uM
NVP-BHG712 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
-16.5
 0.05
uM
NVP-BHG712 PC-3 MAP3K5
DIkGDNVLINTYSGVLK
Lys2
8.9
 0.05
uM
NVP-BHG712 PC-3 MAP3K5,MAP3K6
IAIkEIPER
Lys1
-0.1
 0.05
uM
NVP-BHG712 PC-3 MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
-9.3
 0.05
uM
NVP-BHG712 PC-3 MARK2
EVAVkIIDKTQLNSSSLQK
Lys1
-7.7
 0.05
uM
NVP-BHG712 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
-6.7
 0.05
uM
NVP-BHG712 PC-3 MARK3
EVAIkIIDKTQLNPTSLQK
Lys1
-6.9
 0.05
uM
NVP-BHG712 PC-3 MARK3,MARK4
EVAIkIIDK
Lys1
-13.2
 0.05
uM
NVP-BHG712 PC-3 MAST1,MAST2
DLkPDNLLITSMGHIK
Lys2
-22.3
 0.05
uM
NVP-BHG712 PC-3 MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
3.6
 0.05
uM
NVP-BHG712 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
-3.3
 0.05
uM
NVP-BHG712 PC-3 MASTL
GAFGkVYLGQK
ATP Loop
-1.0
 0.05
uM
NVP-BHG712 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
18.3
 0.05
uM
NVP-BHG712 PC-3 MLK1,MLKL
DLkSSNILILQK
Lys2
-1.3
 0.05
uM