NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 GCN2
LDGCCYAVkR
Lys1
13.3
 0.05
uM
NVP-BHG712 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
-1.8
 0.05
uM
NVP-BHG712 PC-3 GSK3A
DIkPQNLLVDPDTAVLK
Lys2
6.8
 0.05
uM
NVP-BHG712 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
5.4
 0.05
uM
NVP-BHG712 PC-3 ERBB2
GIWIPDGENVKIPVAIkVLR
Lys1
-22.5
 0.05
uM
NVP-BHG712 PC-3 IKKA
DLkPENIVLQDVGGK
Lys2
11.4
 0.05
uM
NVP-BHG712 PC-3 IKKB
DLkPENIVLQQGEQR
Lys2
-1.6
 0.05
uM
NVP-BHG712 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
-14.8
 0.05
uM
NVP-BHG712 PC-3 ILK
WQGNDIVVkVLK
Lys1
-3.2
 0.05
uM
NVP-BHG712 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
-8.2
 0.05
uM
NVP-BHG712 PC-3 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
-18.6
 0.05
uM
NVP-BHG712 PC-3 IRAK4
DIkSANILLDEAFTAK
Lys2
-1.9
 0.05
uM
NVP-BHG712 PC-3 IRE1
DLkPHNILISMPNAHGK
Lys2
5.4
 0.05
uM
NVP-BHG712 PC-3 ITPK1
ESIFFNSHNVSkPESSSVLTELDKIEGVFERPSDEVIR
ATP
-11.7
 0.05
uM
NVP-BHG712 PC-3 JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
-15.8
 0.05
uM
NVP-BHG712 PC-3 JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
0.1
 0.05
uM
NVP-BHG712 PC-3 JAK1 domain2
IGDFGLTkAIETDKEYYTVKDDR
Activation Loop
5.7
 0.05
uM
NVP-BHG712 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
-8.1
 0.05
uM
NVP-BHG712 PC-3 KHS1
NVHTGELAAVkIIK
Lys1
-2.9
 0.05
uM
NVP-BHG712 PC-3 M4K3
NVNTGELAAIkVIK
Lys1
8.1
 0.05
uM
NVP-BHG712 PC-3 LATS1
ALYATkTLR
Lys1
-3.2
 0.05
uM
NVP-BHG712 PC-3 LATS2
DIkPDNILIDLDGHIK
Lys2
-18.0
 0.05
uM
NVP-BHG712 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
0.2
 0.05
uM
NVP-BHG712 PC-3 LOK
NKETGALAAAkVIETK
Lys1
1.8
 0.05
uM
NVP-BHG712 PC-3 LOK
DLkAGNVLMTLEGDIR
Lys2
2.8
 0.05
uM