XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | 91.3 | 10 | uM |
XMD-12 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 10 | uM | |
XMD-12 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -20.1 | 10 | uM |
XMD-12 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -7.5 | 10 | uM |
XMD-12 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -11.7 | 10 | uM |
XMD-12 | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | 10 | uM | |
XMD-12 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | 2.8 | 10 | uM |
XMD-12 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -11.9 | 10 | uM |
XMD-12 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | -10.1 | 10 | uM |
XMD-12 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | 11.4 | 10 | uM |
XMD-12 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 15.8 | 10 | uM |
XMD-12 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 22.4 | 10 | uM |
XMD-12 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -7.1 | 10 | uM |
XMD-12 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | -4.3 | 10 | uM |
XMD-12 | HeLa | BTK | GQYDVAIkMIK | Lys1 | 28.3 | 10 | uM |
XMD-12 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -29.5 | 10 | uM |
XMD-12 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 12.5 | 10 | uM |
XMD-12 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | 14.9 | 10 | uM |
XMD-12 | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 17.6 | 10 | uM |
XMD-12 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 29.7 | 10 | uM |
XMD-12 | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | 5.9 | 10 | uM |
XMD-12 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 51.7 | 10 | uM |
XMD-12 | HeLa | FES | LRADNTLVAVkSCR | Lys1 | -2.5 | 10 | uM |
XMD-12 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | 69.0 | 10 | uM |
XMD-12 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | 14.6 | 10 | uM |