XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | 28.6 | 10 | uM |
| XMD-12 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 36.3 | 10 | uM |
| XMD-12 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | 3.4 | 10 | uM |
| XMD-12 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -17.2 | 10 | uM |
| XMD-12 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -24.3 | 10 | uM |
| XMD-12 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | -31.6 | 10 | uM |
| XMD-12 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -7.5 | 10 | uM |
| XMD-12 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | -26.4 | 10 | uM |
| XMD-12 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -5.2 | 10 | uM |
| XMD-12 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 3.4 | 10 | uM |
| XMD-12 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -12.6 | 10 | uM |
| XMD-12 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -10.2 | 10 | uM |
| XMD-12 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -7.1 | 10 | uM |
| XMD-12 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 14.0 | 10 | uM |
| XMD-12 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -1.6 | 10 | uM |
| XMD-12 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -8.0 | 10 | uM |
| XMD-12 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -11.1 | 10 | uM |
| XMD-12 | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -37.3 | 10 | uM |
| XMD-12 | PC-3 | CDK14 | LVALkVIR | Lys1 | 1.1 | 10 | uM |
| XMD-12 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 1.9 | 10 | uM |
| XMD-12 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 23.7 | 10 | uM |
| XMD-12 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 33.9 | 10 | uM |
| XMD-12 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -5.8 | 10 | uM |
| XMD-12 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.2 | 10 | uM |
| XMD-12 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 26.6 | 10 | uM |