XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | PC-3 | MAP2K6 | HVPSGQIMAVkR | Lys1 | 23.7 | 10 | uM |
XMD-12 | HeLa | MAP3K1 | DVkGANLLIDSTGQR | Lys2 | 53.5 | 10 | uM |
XMD-12 | PC-3 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 75.4 | 10 | uM |
XMD-12 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | 39.6 | 10 | uM |
XMD-12 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 18.0 | 10 | uM |
XMD-12 | HeLa | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -23.3 | 10 | uM |
XMD-12 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -0.6 | 10 | uM |
XMD-12 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | -13.0 | 10 | uM |
XMD-12 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 38.2 | 10 | uM |
XMD-12 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 72.5 | 10 | uM |
XMD-12 | HeLa | MAST2,MAST4 | DLkPDNLLVTSMGHIK | Lys2 | -4.9 | 10 | uM |
XMD-12 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 8.2 | 10 | uM |
XMD-12 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 15.2 | 10 | uM |
XMD-12 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 21.7 | 10 | uM |
XMD-12 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 40.1 | 10 | uM |
XMD-12 | HeLa | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 93.5 | 10 | uM |
XMD-12 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 81.1 | 10 | uM |
XMD-12 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | 14.4 | 10 | uM |
XMD-12 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -71.5 | 10 | uM |
XMD-12 | HeLa | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 65.3 | 10 | uM |
XMD-12 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 73.5 | 10 | uM |
XMD-12 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | 39.1 | 10 | uM |
XMD-12 | HeLa | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 36.1 | 10 | uM |
XMD-12 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 53.0 | 10 | uM |
XMD-12 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | 15.0 | 10 | uM |