XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 97.4 | 10 | uM |
| XMD-12 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | -9.6 | 10 | uM |
| XMD-12 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 95.0 | 10 | uM |
| XMD-12 | HeLa | PKR | DLkPSNIFLVDTK | Lys2 | -9.5 | 10 | uM |
| XMD-12 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | 94.6 | 10 | uM |
| XMD-12 | HeLa | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 93.5 | 10 | uM |
| XMD-12 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -9.3 | 10 | uM |
| XMD-12 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 92.9 | 10 | uM |
| XMD-12 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.2 | 10 | uM |
| XMD-12 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 91.5 | 10 | uM |
| XMD-12 | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | 91.3 | 10 | uM |
| XMD-12 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 90.3 | 10 | uM |
| XMD-12 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 88.8 | 10 | uM |
| XMD-12 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 88.7 | 10 | uM |
| XMD-12 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -8.8 | 10 | uM |
| XMD-12 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 87.9 | 10 | uM |
| XMD-12 | PC-3 | PITSLRE | DLkTSNLLLSHAGILK | Lys2 | -8.6 | 10 | uM |
| XMD-12 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 85.4 | 10 | uM |
| XMD-12 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.5 | 10 | uM |
| XMD-12 | PC-3 | LOK | NKETGALAAAkVIETK | Lys1 | 84.5 | 10 | uM |
| XMD-12 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | 8.4 | 10 | uM |
| XMD-12 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 8.2 | 10 | uM |
| XMD-12 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 81.3 | 10 | uM |
| XMD-12 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 81.1 | 10 | uM |
| XMD-12 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -8.0 | 10 | uM |