XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 15.0 | 10 | uM |
| XMD-12 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -10.0 | 10 | uM |
| XMD-12 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 30.5 | 10 | uM |
| XMD-12 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 30.6 | 10 | uM |
| XMD-12 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -7.3 | 10 | uM |
| XMD-12 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 88.7 | 10 | uM |
| XMD-12 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -14.1 | 10 | uM |
| XMD-12 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -4.3 | 10 | uM |
| XMD-12 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.2 | 10 | uM |
| XMD-12 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 97.4 | 10 | uM |
| XMD-12 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -16.7 | 10 | uM |
| XMD-12 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.3 | 10 | uM |
| XMD-12 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 70.4 | 10 | uM |
| XMD-12 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 24.9 | 10 | uM |
| XMD-12 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 1.1 | 10 | uM |
| XMD-12 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 88.8 | 10 | uM |
| XMD-12 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -11.3 | 10 | uM |
| XMD-12 | HeLa | ATR | FYIMMCkPK | ATP | -2.1 | 10 | uM |
| XMD-12 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 87.9 | 10 | uM |
| XMD-12 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 62.7 | 10 | uM |
| XMD-12 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -6.9 | 10 | uM |
| XMD-12 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -16.3 | 10 | uM |
| XMD-12 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -16.8 | 10 | uM |
| XMD-12 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 92.9 | 10 | uM |
| XMD-12 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -25.1 | 10 | uM |