XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | -50.1 | 10 | uM |
| XMD8-92 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 7.8 | 10 | uM |
| XMD8-92 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | -20.9 | 10 | uM |
| XMD8-92 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 6.9 | 10 | uM |
| XMD8-92 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 3.4 | 10 | uM |
| XMD8-92 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.5 | 10 | uM |
| XMD8-92 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -5.5 | 10 | uM |
| XMD8-92 | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | -6.2 | 10 | uM |
| XMD8-92 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -18.1 | 10 | uM |
| XMD8-92 | HeLa | TLK1 | YAAVkIHQLNK | Lys1 | 3.0 | 10 | uM |
| XMD8-92 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | 13.2 | 10 | uM |
| XMD8-92 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.9 | 10 | uM |
| XMD8-92 | PC-3 | ILK | WQGNDIVVkVLK | Lys1 | 17.7 | 10 | uM |
| XMD8-92 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | -0.8 | 10 | uM |
| XMD8-92 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 10.9 | 10 | uM |
| XMD8-92 | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -3.4 | 10 | uM |
| XMD8-92 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -16.1 | 10 | uM |
| XMD8-92 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -7.0 | 10 | uM |
| XMD8-92 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | 14.2 | 10 | uM |
| XMD8-92 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 7.0 | 10 | uM |
| XMD8-92 | HeLa | PAN3 | VMDPTkILITGK | -4.5 | 10 | uM | |
| XMD8-92 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -20.2 | 10 | uM |
| XMD8-92 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -4.9 | 10 | uM |
| XMD8-92 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 11.1 | 10 | uM |
| XMD8-92 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -2.0 | 10 | uM |