XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -28.7 | 10 | uM |
| XMD8-92 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 40.4 | 10 | uM |
| XMD8-92 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -18.4 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
| XMD8-92 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.7 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 6.7 | 10 | uM |
| XMD8-92 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 3.9 | 10 | uM |
| XMD8-92 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | 10.0 | 10 | uM |
| XMD8-92 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -15.6 | 10 | uM |
| XMD8-92 | PC-3 | ATR | FYIMMCkPK | ATP | 6.1 | 10 | uM |
| XMD8-92 | HeLa | ATR | FYIMMCkPK | ATP | -5.7 | 10 | uM |
| XMD8-92 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 9.7 | 10 | uM |
| XMD8-92 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 9.3 | 10 | uM |
| XMD8-92 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -15.5 | 10 | uM |
| XMD8-92 | HeLa | BTK | GQYDVAIkMIK | Lys1 | -9.2 | 10 | uM |
| XMD8-92 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -6.3 | 10 | uM |
| XMD8-92 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -3.6 | 10 | uM |
| XMD8-92 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 18.5 | 10 | uM |
| XMD8-92 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 7.2 | 10 | uM |
| XMD8-92 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 2.7 | 10 | uM |
| XMD8-92 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 1.6 | 10 | uM |
| XMD8-92 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | -8.1 | 10 | uM |
| XMD8-92 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 2.8 | 10 | uM |
| XMD8-92 | PC-3 | CDK14 | LVALkVIR | Lys1 | -6.6 | 10 | uM |
| XMD8-92 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 17.9 | 10 | uM |